Noopept (157115-85-0) - Cofttek

Noopept (157115-85-0)

Nwere ike 7, 2021

Cofttek bụ onye nrụpụta ntụ ntụ Noopept kacha mma na China. Ụlọ ọrụ anyị nwere zuru ezu mmepụta usoro njikwa (ISO9001 & ISO14001), na ikike mmepụta kwa ọnwa nke 600kg.

 


ọnọdụ:Na Production Production
Otu:1kg / akpa, 25kg / Drum

Noopept (157115-85-0) Smmezi

aha:Noopept
CAS:157115-85-0
ọcha98%
Usoro Molecular:C17H22N2O4
Molekụla arọ:318.37 g / moll
Melt Point:94.0 ka 98.0 Celsius C
Aha aha:ethyl 2-[[(2S)-1-(2-phenylacetyl)pyrrolidine-2-carbonyl]amino]acetate
Synonyms:Noopept; ethyl 2 - [[(2S) -1- (2-phenylacetyl) pyrrolidine-2-carbonyl] amino] acetate; N- (1- (Phenylacetyl) -L-prolyl) glycine ethyl ester; Ethyl 1- (phenylacetyl) ) -L-prolylglycinate; noopept ntụ ntụ; Nootropic GVS-111; (S) -ethyl 2- (1- (2-phenylacetyl) pyrrolidine-2-carboxaMido) acetate; SGS 111
KeyInChI:PJNSMUBMSNAEEN-AWEZNQCLSA-N
Ọkara ndụ:Noopept ọkara ndụ bụ naanị 60 ruo 90 nkeji, nke pụtara na mmadụ nkịtị nwere ike ịhazi ọkara nke ọgwụ ahụ n'oge ahụ.
Solubility:Soluble na DMSO (25 mg / ml)
Ọnọdụ Nchekwa:0 - 4 C maka obere oge (ụbọchị ruo izu), ma ọ bụ -20 C maka ogologo oge (ọnwa)
ngwa:Noopept bụ ihe na-ewu ewu na-akwalite ọgụgụ isi mgbakwunye na nootropic obodo. Ọmụmụ mmadụ egosila nsonaazụ na-ekwe nkwa, yana ngwa nwere ike na ọgwụgwọ ọrịa Alzheimer.
anya:ọcha ka beige ntụ ntụ

 

Gịnị bụ Noopept (157115-85-0)?

Noopept bụ aha aha maka N-phenylacetyl-L-prolylglycine ethyl ester; ihe na-emepụta ihe nootropic na-ekwukarị na ọ bụ akụkụ nke òtù racetam nke nootropics (ọ nweghị oghere 2-oxo-pyrollidine nke mere na ọ bụghị racetam). Na Russia, ebe eburu aha ya bụ Noopept, mgbe ụfọdụ a na-akpọ ya GSV-111.

E kere Noopept na 1996. Ihe owuwu ya dabere na nke cycloprolylglycine; ihe omimi neuropeptide. A maara Cycloprolylglycine iji kwalite okwu nke Brain Na-enweta Neurotrophic Factor na ụbụrụ. Ndị nchọpụta mere ka ọ bụrụ na nootropic dabere na cycloprolylglycine ga-enwe mmetụta yiri nke ahụ, nke ahụ bụ kpọmkwem ihe a na-ekwu banyere Noopept.

Ọ bụ ezie na ọ bụghị racetam, Noopept yiri nke Piracetam. Noopept bụ n'ezie dipeptide conjugate nke Piracetam. A na-ekwu na mkpụrụ ndụ abụọ ahụ nwere mmetụta yiri nke ahụ, na Noopept bụ ikike dị ukwuu nke nootropics abụọ ahụ site na ibu.

 

Noopept (157115-85-0) uru

Uru ndị metụtara Noopept dị ọtụtụ ma dịgasị iche iche. Nke a abụghị ihe mgbagwoju anya nyere ya na ọ nwere ike ịme acetylcholine ma na-abawanye ogo nke NGF na BDNF.

Nke a bụ ndepụta nke uru ndị metụtara Noopept:

  • Nchekwa ka mma ọrụ
  • Enwekwukwa anya, ilekwasị anya na itinye uche
  • Mụ anya ịmụ anya
  • Na-akwalite nhụjuanya na uto nke ụbụrụ ụbụrụ ọhụrụ
  • Na-ebelata nrụgide oxidative ma na-akwalite ahụike ụbụrụ
  • Belata nchekasị ma na-akwalite excitability

Ihe ndị a niile ga-esi na ọnụọgụ nnabata acetylcholine na-arịwanye elu na akpụkpọ anụ neuronal yana site na ịba ụba NGF / BDNF n'ogologo. Mmetụta nke ibuli neuropeptide nwere na cognition dị egwu, ọ ga-ahụkwa mmetụta dị mkpirikpi nke ike nke acetylcholine. Nchịkọta nke usoro abụọ a ga-abụ njikarịcha ụbụrụ zuru oke, yana akụkụ ọ bụla nke ụbụrụ na-arụ ọrụ n'ụzọ ka mma n'ụzọ ụfọdụ.

 

Noopept (157115-85-0) jiri?

Noopept bụ ihe mgbakwunye na-ewu ewu na-eme ka enwe mmetụta na obodo nootropic. A na-eji Noopept eme ihe maka ịbawanye akara acetylcholine, na-amụba okwu nke BDNF na NGF, na-echebe site na ịba ụba glutamate, na ịba ụba na-egbochi ụbụrụ na ụbụrụ. Ihe ndi a bu ihe eji eme ihe bu ihe omumu.

 

Noopept (157115-85-0) Ọgwụ

Ngwunye noopept nwere ike ịbụ ihe mgbagwoju anya, ọkachasị maka ndị mbido, mana nke a bụ ngwa ngwa ma dịkwa mfe iji nyere gị aka ịpụ.

Cheta, mgbe Noopept na-tụnyere Piracetam, ọ bụ n'ezie ruo 1000 ugboro ike karịa Piracetam!

Na na kwuru, adịghị eji otu ego na ị ga-ejikari ime Piracetam ma ọ bụ ọbụna na ndị ọzọ nootropics na yiri mmetụta.

Dị ka iwu zuru oke, ị ga-agbasakwa otu ọgwụ ụbọchị niile ma were ezumike mgbe ọ bụla ọnwa abụọ maka ebumnuche nchekwa.

 

  • Oral Dosage

Ngwadogwu akwadoro maka okenye bụ 10-30 mg, dabere na ibu gị. Agbanyeghị, ọ kachasị mma ịmalite site na naanị 10 mg iji chọpụta mmetụta dị na ahụ gị.

A sị ka e kwuwe, ịnwere ike ị increaseụ ọgwụ ahụ mgbe niile.

Capsules nwere nha dịgasị iche, yabụ kpachara anya ịlele akara ahụ nke ọma tupu ịzụrụ karama.

Were naanị obere ego ịchọrọ maka nchekwa gị. Nke a ga - enye aka gbochie gị ịmebe ọgwụ.

 

  • Lingdị Ọgwụ Nke Abụọ

Maka usoro onunu ogwu, ikwesiri ibido ntakịrị, na gburugburu 5 mg.

Ebe ọ bụ na ọ nwere nsonaazụ ngwa ngwa ma sie ike karị, ị kwesịrị ịlele etu ị si meghachi omume na usoro a tupu ịbawanye ogo 10 mg.

Ọ dị ezigbo mkpa ịlele nha ntụ ntụ nke ịchọrọ. Ọgwụ dị elu nwere ike ibute Noopept nsogbu mmetụta, yabụ kpachara anya!

 

Yiri usoro onunu ogwu, ogwu ogwu nke ogwu kwesiri idi ala.

Ọ bụ ezie na ọ dị mma iji 10-30 mg n'ụdị ọ bụla, Noopept nwere ike ibute isi ọwụwa, ike ọgwụgwụ na ọgbụgbọ, yabụ na-emehie mgbe niile.

 

  • Megadose

Ọ bụrụ na ụdị ọgwụ dị na 10 ruo 30 milligrams, Noopept megadose bụ onye na-egbu 50 ka 100 milligram. Fọdụ ndị mmadụ na-ewere ihe karịrị 100 mg!

A na-eji megadose mee ihe mgbe ịchọrọ ịhụ ihe dị egwu nkwalite na ebe nchekwa gị, mmụta, ọgụgụ isi, na n'ozuzu nka nka.

A ga-eme nke a otu ugboro n'izu kachasị, n'ihi na iji ya eme ihe nwere ike ime ka ọ ghara ịdị irè na ogologo oge.

Tụkwasị na nke a, nke a nwere ike ịdị oke egwu nye ụfọdụ ndị, yabụ gbaa mbọ hụ na ị maara nke ọma ogo ndidi gị tupu ịnwale nke a.

 

Noopept ntụ ntụ n'ihi na ire (Ebe ịzụta Noopept ntụ ntụ na nnukwu)

Ụlọ ọrụ anyị na-enwe mmekọrịta ogologo oge na ndị ahịa anyị n'ihi na anyị na-elekwasị anya na ndị ahịa ọrụ na inye nnukwu ngwaahịa. Ọ bụrụ na i nwere mmasị na anyị ngwaahịa, anyị na-agbanwe na customization nke iwu ona gị kpọmkwem mkpa na anyị ngwa ngwa ụzọ oge na iwu emesi ị ga-enwe oké akatabi okop ngwaahịa anyị na-oge. Anyị na-elekwasịkwa anya na ọrụ ndị bara uru. Anyị dị maka ajụjụ ọrụ na ozi iji kwado azụmahịa gị.

Anyị bụ ndị ọkachamara Noopept ntụ ntụ soplaya ruo ọtụtụ afọ, anyị na-enye ngwaahịa na ọnụahịa asọmpi, na ngwaahịa anyị bụ nke kachasị mma ma na-enweta nnwale siri ike, nke onwe ya iji hụ na ọ dị mma maka oriri gburugburu ụwa.

 

References

[1] Ostrovskaya RU, Gudasheva TA, Zaplina AP, Vahitova JV, Salimgareeva MH, Jamidanov RS, Seredenin SB. Noopept na-akpali okwu nke NGF na BDNF na rat hippocampus. Bull Exp Biol Ahụike. 2008 Sep; 146 (3): 334-7. ma ọ bụ: 10.1007 / s10517-008-0297-x. PMID: 19240853.

[2] Neznamov GG, Teleshova ES. Ntụnyere ọmụmụ nke Noopept na piracetam na ọgwụgwọ nke ndị ọrịa na-enwe nsogbu nghọta dị nro na ọrịa ụbụrụ ụbụrụ nke ọrịa vaskụla na traumatic sitere. Neurosci Behav Physiol. 2009 Maachị; 39 (3): 311-21 . doi: 10.1007/s11055-009-9128-4. PMID: 19234797.

[3] Murzina, GB, Pivovarov, AS Modulation nke Acetylcholine-Ntinye Ntinye Ugbu a site na Noopept na Helix Lucorum Neurons. BIOPHYSICS 64, 393–399 (2019).

[4] Neznamov, GG; Teleshova, ES (2009). "Comparative ọmụmụ Noopept na piracetam na ọgwụgwọ nke ndị ọrịa nwere nwayọọ cognitive ọrịa na organic ụbụrụ ọrịa nke vaskụla na traumatic si malite". Neuroscience na Ahụhụ Ahụhụ. 39 (3): 311–321.

[5] Tardner, P (2020). "Findchọta ezigbo onunu ogwu fornootropic agent Noopept: Nchoputa nke akwukwo di" (PDF). International Journal of Environmental Science na Teknụzụ.

 


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